Improved synthesis of 2-amino-1, 2, 4-triazolo [1, 5-a] pyrimidines

VM Chernyshev, AN Sokolov…

Index: Chernyshev; Sokolov; Taranushich Russian Journal of Applied Chemistry, 2006 , vol. 79, # 7 p. 1134 - 1137

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Citation Number: 10

Abstract

Abstract An improved procedure is suggested for preparing 2-amino-1, 2, 4-triazolo [1, 5-a] pyrimidines from 3, 5-diamino-1, 2, 4-triazole and unsaturated aromatic ketones, with acetyl protection of the amino group in the step of oxidation of 2-amino-4, 7-dihydro-1, 2, 4-triazolo [1, 5-a] pyrimidines.