LG 82-4-01

Names

[ Name ]:
LG 82-4-01

[Synonym ]:
LG 82-4-01
4-chloro-5-[2-(1h-imidazol-1-yl)ethoxy]thiophene-2-carboxylic acid hydrochloride(1:1)
5-(2-(1-Imidazolyl)ethoxy)-4-chlorothiophene-2-carboxylic acid

Biological Activity

[Description]:

LG 82-4-01 is a thromboxane (TX) synthetase specific inhibitor, with an IC50 of 1.3 μM[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Prostaglandin Receptor

Research Areas >> Metabolic Disease

[References]

[1]. E F Smith 3rd, et al. Inhibition of thromboxane and 12-HPETE formation by dazoxiben and its two thiophenic acid-substituted derivatives. Eur J Pharmacol. 1985 Jun 7;112(2):161-9.

Chemical & Physical Properties

[ Boiling Point ]:
540.6ºC at 760mmHg

[ Molecular Formula ]:
C₁₀H₁₀Cl₂N₂O₃S

[ Molecular Weight ]:
309.16900

[ Flash Point ]:
280.8ºC

[ Exact Mass ]:
307.97900

[ PSA ]:
92.59000

[ LogP ]:
3.17720

LG 82-4-01

Names

Biological Activity

Chemical & Physical Properties

Related Compounds