TAK-100
Names
[ CAS No. ]:
907609-33-0
[ Name ]:
TAK-100
Biological Activity
[Description]:
TAK-100 is a potent, selective and orally active inhibitor of DPP-4 with IC50 of 5.3 nM, shows no inhibition on DPP2/8/9. Diabetes Phase 1 Discontinued
[References]
References 1. Miyamoto Y, et al. J Med Chem. 2011 Feb 10;54(3):831-50. View Related Products by Target Dipeptidyl Peptidase (DPP) Diabetes
Chemical & Physical Properties
[ Molecular Formula ]:
C22H30N2O2
[ Molecular Weight ]:
354.494