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Darenzepine

Names

[ CAS No. ]:
84629-61-8

[ Name ]:
Darenzepine

[Synonym ]:
Darenzepine
11H-Dibenz[b,e]azepine, piperazine deriv.
DARENZEPINE
Piperazine, 1-[(5,6-dihydro-6-oxo-11H-dibenz[b,e]azepin-11-ylidene)acetyl]-4-methyl-, (E)-

Biological Activity

[Description]:

Darenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> mAChR
Signaling Pathways >> Neuronal Signaling >> mAChR
Research Areas >> Neurological Disease

[Target]

muscarinic receptor[1]


[In Vitro]

Darenzepine is a muscarinic receptor inhibitor which is useful for the treatment of CNS disorders[1].

[References]

[1]. Eric Elenko, et al. Methods and compositions for treatment of disorders ameliorated by muscarinic receptor activation. US 20170095465 A1.


[Related Small Molecules]

Carbachol | Darifenacin HBr | Arecoline hydrobromide | Pirenzepine, Dihydrochloride | Glycopyrrolate | Imidafenacin | Benztropine Mesylate | Xanomeline oxalate | Batefenterol | Bethanechol chloride | Cevimeline hydrochloride hemihydrate | Otilonium Bromide | solifenacin | VU0467154 | Anisodamine

Chemical & Physical Properties

[ Molecular Formula ]:
C21H21N3O2

[ Molecular Weight ]:
347.41000

[ Exact Mass ]:
347.16300

[ PSA ]:
56.41000

[ LogP ]:
1.39270

[ Storage condition ]:
2-8℃

Related Compounds