MEK1 Derived Peptide Inhibitor 1

Names

[ CAS No. ]:
355367-87-2

[ Name ]:
MEK1 Derived Peptide Inhibitor 1

Biological Activity

[Description]:

MEK1 Derived Peptide Inhibitor 1 is a peptide inhibitor. MEK1 Derived Peptide Inhibitor 1 can inhibit the in vitro activation of ERK2 by MEK1 with an IC50 value of 30 μM. MEK1 Derived Peptide Inhibitor 1 can be used for the research of cell-permeable[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> MAPK/ERK Pathway >> MEK
Signaling Pathways >> MAPK/ERK Pathway >> ERK
Signaling Pathways >> Stem Cell/Wnt >> ERK

[References]

[1]. Bradley R Kelemen, et al. Selective in vivo inhibition of mitogen-activated protein kinase activation using cell-permeable peptides. J Biol Chem. 2002 Mar 8;277(10):8741-8.  

Chemical & Physical Properties

[ Molecular Formula ]:
C68H118N18O17S

[ Molecular Weight ]:
1491.84

Related Compounds