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CBP/P300 bromodomain inhibitor-3

Names

[ CAS No. ]:
2304416-91-7

[ Name ]:
CBP/P300 bromodomain inhibitor-3

Biological Activity

[Description]:

CBP/P300 bromodomain inhibitor-3 is a potent inhibitor of the CBP/P300 family of bromodomains. CBP/P300 bromodomain inhibitor-3 inhibits CBP (IC50=0.01-0.1 µΜ) and BRD4 (IC50=1-1000 µΜ) activity[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[Target]

BRD4:1-1000 μM (IC50)

CBP:0.01-0.1 μM (IC50)


[References]

[1]. Shawn E.R. Schiller, et al. Tetrahydro-imidazo quinoline compositions as cbp/p300 inhibitors. WO2019055877A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C27H31N3O4

[ Molecular Weight ]:
461.55

Related Compounds