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ATX inhibitor 1

Names

[ CAS No. ]:
2225892-70-4

[ Name ]:
ATX inhibitor 1

Biological Activity

[Description]:

ATX inhibitor 1 is a potent ATX (IC50=1.23 nM, FS-3 and 2.18 nM, bis-pNPP) inhibitor.

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Phosphodiesterase (PDE)
Research Areas >> Others

[Target]

IC50: 1.23 nM (FS-3) and 2.18 nM (bis-pNPP)[1]


[References]

[1]. Balupuri A, et al. Discovery and optimization of ATX inhibitors via modeling, synthesis and biological evaluation. Eur J Med Chem. 2018 Mar 25;148:397-409.

Chemical & Physical Properties

[ Molecular Formula ]:
C21H23Cl2N2O6P

[ Molecular Weight ]:
501.30

Related Compounds