Cavα2δ1&NET-IN-3

Names

[ CAS No. ]:
2143584-82-9

[ Name ]:
Cavα2δ1&NET-IN-3

Biological Activity

[Description]:

Cavα2δ1&NET-IN-3 (example 216) is an inhibitor of the subunit α2δ of voltage-gated calcium channels (VGCC) and noradrenaline transporter (NET). Cavα2δ1&NET-IN-3 has Kis of 100-500 nM for human α2δ-1 subunit of Cav2.2 calcium channel and NET, respectively[1].

[Related Catalog]:

Signaling Pathways >> Membrane Transporter/Ion Channel >> Calcium Channel
Research Areas >> Endocrinology
Research Areas >> Neurological Disease

[Target]

Calcium Channel


[References]

[1]. subunit α2δ of voltage-gated calcium channels (VGCC) and noradrenaline transporter (NET). Cavα2δ1&NET-IN-3 has kis of 100-500 nM for human α2δ-1 subunit of Cav2.2

Chemical & Physical Properties

[ Molecular Formula ]:
C24H30N6O2S

[ Molecular Weight ]:
466.60

Related Compounds