PCSK9-IN-2

Names

[ CAS No. ]:
2099167-44-7

[ Name ]:
PCSK9-IN-2

Biological Activity

[Description]:

PCSK9-IN-2 is a novel small molecule inhibitor of PCSK9-LDLR protein–protein interaction (PPI) with an IC50 value of 7.57 μM.

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Ser/Thr Protease

Research Areas >> Cardiovascular Disease

[References]

[1]. Sun H, et al. Discovery of Novel Small Molecule Inhibitors Disrupting the PCSK9-LDLR Interaction. J Chem Inf Model. 2021 Oct 25;61(10):5269-5279.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₆H₃₂N₆O₆

[ Molecular Weight ]:
524.57

Related Compounds

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