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Mitapivat

Names

[ CAS No. ]:
1260075-17-9

[ Name ]:
Mitapivat

[Synonym ]:
PKM2 activator 1020
Mitapivat

Biological Activity

[Description]:

Mitapivat is a potent human R-type pyruvate kinase (PKR) inhibitor; also shows potency for mutant PKR including R510Q PKR, R532W PKR, T384W PKR etc.

[Related Catalog]:

Signaling Pathways >> Others >> Others
Research Areas >> Cancer

[References]

[1]. PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY. Patent WO/2012/151451A1


[Related Small Molecules]

Captisol | Cyclosporin A | H2DCFDA | 0MPTP hydrochloride | GW4869 | Etomoxir | TD139 | Mitoquinone mesylate | GSK2795039 | JC-1 | BAPTA-AM | AP 20187 | Setanaxib (GKT137831) | D-Luciferin | Crotaline

Chemical & Physical Properties

[ Molecular Formula ]:
C24H26N4O3S

[ Molecular Weight ]:
450.55300

[ Exact Mass ]:
450.17300

[ PSA ]:
90.99000

[ LogP ]:
4.23300

Related Compounds

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