GPR81 agonist 2

Names

[ CAS No. ]:
1143024-28-5

[ Name ]:
GPR81 agonist 2

Biological Activity

[Description]:

GPR81 agonist 2 (compound 1) is a potent GPR81 agonist with EC50 values of 0.023, 0.123 µM for hGPR81, hGPR109A, respectively[1].

[Related Catalog]:

Signaling Pathways >> Others >> Others
Research Areas >> Metabolic Disease

[Target]

EC50: 0.023 (hGPR81); 0.123 µM (hGPR109A)[1]


[References]

[1]. Davidsson Ö, et al. Identification of novel GPR81 agonist lead series for target biology evaluation. Bioorg Med Chem Lett. 2020 Feb 15;30(4):126953.  

Chemical & Physical Properties

[ Molecular Formula ]:
C26H27ClN6O5S2

[ Molecular Weight ]:
603.11

Related Compounds